SCHEMBL8948031

SCHEMBL8948031

O=c1[nH]c2ccc(CCCCN3CCOCC3)cc2o1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.49
DRD2 P14416 1/20 0.49
HTR2A P28223 1/20 0.49
SLC6A2 P23975 1/20 0.49
SLC6A3 Q01959 1/20 0.49
SIGMAR1 Q99720 4/20 0.45
POLB P06746 1/20 0.45
GRIN1 Q05586 3/20 0.43
GRIN2D O15399 2/20 0.43
GRIN3B O60391 2/20 0.43
GRIN2A Q12879 2/20 0.43
GRIN2B Q13224 2/20 0.43
GRIN2C Q14957 2/20 0.43
GRIN3A Q8TCU5 2/20 0.43
LSS P48449 1/20 0.43
PARP1 P09874 2/20 0.42
TSHR P16473 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NOS1 P29475 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9463759 0.96 HTR1A (0.50) HTR1ADRD2HTR2ASLC6A2SLC6A3
Hydrochloric Acid SCHEMBL9464214 0.95 HTR1A (0.49) HTR1ADRD2HTR2ASLC6A2SLC6A3
SCHEMBL9463689 0.86 HTR1A (0.52) HTR1ADRD2HTR2ASLC6A2SLC6A3
SCHEMBL9464172 0.85 HTR1A (0.51) HTR1ADRD2HTR2ASLC6A2SLC6A3
SCHEMBL9465050 0.84 HTR1A (0.55) HTR1ADRD2HTR2ASLC6A2SLC6A3
SCHEMBL10394028 0.81 DRD2 (0.62) HTR1ADRD2HTR2ASLC6A2SLC6A3
SCHEMBL8109444 0.81 SIGMAR1 (0.58) DRD2SIGMAR1GRIN1TSHRMEN1
SCHEMBL8100582 0.80 GRIN1 (0.66) SIGMAR1GRIN1GRIN2DGRIN3BGRIN2A
SCHEMBL10393591 0.80 HTR1A (0.59) HTR1ADRD2HTR2ASLC6A2SLC6A3
SCHEMBL9463532 0.79 HTR1A (0.48) HTR1ADRD2HTR2ASLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed