SCHEMBL8948066

SCHEMBL8948066

O=c1[nH]c2ccc(CCN3CCN(c4cccnc4)CC3)cc2s1

nearest known ligand 0.77

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 13/20 0.77
HTR2C P28335 8/20 0.77
DRD2 P14416 4/20 0.58
HTR2A P28223 4/20 0.58
DRD4 P21917 1/20 0.47
HTR7 P34969 1/20 0.47
DRD3 P35462 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948209 0.87 HTR1A (1.00) HTR1AHTR2CDRD2HTR2A
SCHEMBL8786139 0.83 HTR1A (0.72) HTR1AHTR2CDRD2HTR2ADRD4
SCHEMBL8785477 0.81 HTR1A (0.79) HTR1AHTR2CDRD2HTR2ADRD3
SCHEMBL8948002 0.81 HTR1A (0.87) HTR1AHTR2CDRD2HTR2AHTR7
SCHEMBL9449656 0.80 HTR1A (0.77) HTR1AHTR2C
SCHEMBL8947912 0.80 HTR1A (0.85) HTR1AHTR2CDRD2HTR2AHTR7
SCHEMBL8785701 0.80 HTR1A (1.00) HTR1AHTR2CDRD2HTR2ADRD3
SCHEMBL4891426 0.75 HTR1A (0.75) HTR1AHTR2CDRD2HTR2A
SCHEMBL8786294 0.75 HTR1A (1.00) HTR1AHTR2CDRD2HTR2A
SCHEMBL8948219 0.75 HTR1A (0.70) HTR1AHTR2CDRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed