SCHEMBL8947935

SCHEMBL8947935

O=C(c1ccc(F)cc1)C1CCN(CCn2c(=O)sc3cc(CCN4CCOCC4)ccc32)CC1

nearest known ligand 0.89

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.59
HTR2C P28335 3/20 0.59
HTR7 P34969 3/20 0.59
HTR6 P50406 3/20 0.59
HTR1A P08908 1/20 0.52
TMEM97 Q5BJF2 1/20 0.49
SIGMAR1 Q99720 2/20 0.48
ADRA2A P08913 1/20 0.48
ADRA2B P18089 1/20 0.48
ADRA2C P18825 1/20 0.48
HRH1 P35367 1/20 0.48
KCNH2 Q12809 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948078 0.94 HTR2A (0.55) HTR2AHTR2CHTR7HTR6TMEM97
SCHEMBL8947898 0.92 HTR2A (0.55) HTR2AHTR2CHTR7HTR6SIGMAR1
SCHEMBL8948011 0.89 HTR1A (0.60) HTR2AHTR2CHTR7HTR6HTR1A
SCHEMBL8947974 0.89 SIGMAR1 (0.64) HTR2AHTR2CHTR7HTR6SIGMAR1
SCHEMBL8948007 0.87 HTR1A (0.66) HTR2AHTR2CHTR7HTR6HTR1A
SCHEMBL8947902 0.85 KCNH2 (0.53) TMEM97SIGMAR1KCNH2
SCHEMBL8947787 0.85 SIGMAR1 (0.58) HTR2ATMEM97SIGMAR1
SCHEMBL8948106 0.85 HTR2A (0.49) HTR2AHTR2CHTR7HTR6HTR1A
SCHEMBL8948101 0.85 TMEM97 (0.49) HTR1ATMEM97SIGMAR1
SCHEMBL8948061 0.85 SIGMAR1 (0.52) HTR2AHTR2CHTR7HTR6TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed