SCHEMBL8948221

SCHEMBL8948221

O=C(c1ccc(F)cc1)C1CCN(CCCCc2ccc3[nH]c(=O)oc3c2)CC1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.61
KDM4E B2RXH2 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2D6 P10635 1/20 0.61
GRIN2D O15399 2/20 0.60
GRIN3B O60391 2/20 0.60
GRIN1 Q05586 2/20 0.60
GRIN2A Q12879 2/20 0.60
GRIN2B Q13224 2/20 0.60
GRIN2C Q14957 2/20 0.60
GRIN3A Q8TCU5 2/20 0.60
HTR2C P28335 3/20 0.56
HTR7 P34969 3/20 0.56
HTR6 P50406 3/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947923 0.91 KCNH2 (0.56) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL8947955 0.91 HTR2A (0.55) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9161222 0.88 LMNA (0.47) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL8948079 0.82 HTR2A (0.62) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL4675791 0.82 GRIN1 (0.71) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL8948109 0.81 HTR2A (0.61) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL8947873 0.78 HTR2A (0.56) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL10393591 0.77 HTR1A (0.59) HTR2AGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8109942 0.77 GRIN1 (0.74) HTR2AGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8109444 0.77 SIGMAR1 (0.58) CYP1A2CYP3A4CYP2D6GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed