SCHEMBL8948496

SCHEMBL8948496

CC(C)(C)OC(=O)C1CCN(CC2CN(c3ccc(NC(=N)N)cc3)C(=O)O2)CC1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.47
ITGA2B P08514 10/20 0.47
PRSS1 P07477 9/20 0.47
PRSS2 P07478 9/20 0.47
PRSS3 P35030 9/20 0.47
F10 P00742 9/20 0.46
SIGMAR1 Q99720 7/20 0.43
F2 P00734 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948623 0.88 SIGMAR1 (0.48) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8316698 0.88 ITGB3 (0.43) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8313822 0.86 ITGB3 (0.54) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8948804 0.85 SIGMAR1 (0.46) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8948666 0.83 GRM2 (0.49) ITGB3ITGA2BSIGMAR1
SCHEMBL8948671 0.83 GRM2 (0.49) ITGB3ITGA2BSIGMAR1
SCHEMBL8948655 0.82 SIGMAR1 (0.44) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8313827 0.81 ITGB3 (0.45) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8948761 0.77 ITGB3 (0.72) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8948798 0.77 ITGB3 (0.72) ITGB3ITGA2BPRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1052231-C Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2000-05-10 CN disclosed
US-5532255-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-07-02 US disclosed
CN-1097421-A Adhesion receptor antagonists MERCK PATENT GMBH (DE) 1995-01-18 CN disclosed