SCHEMBL8948759

SCHEMBL8948759

N#Cc1ccc(N2CC(CN3CCN(CCC(=O)OCc4ccccc4)CC3)OC2=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.45
GRM2 Q14416 7/20 0.44
L3MBTL1 Q9Y468 1/20 0.42
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
HRH1 P35367 3/20 0.41
SLC6A2 P23975 2/20 0.41
HRH2 P25021 2/20 0.41
TMEM97 Q5BJF2 2/20 0.41
CHRM1 P11229 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
HTR1A P08908 2/20 0.40
HTR2A P28223 2/20 0.40
DRD4 P21917 1/20 0.40
OPRM1 P35372 1/20 0.40
CHRM5 P08912 1/20 0.40
ADRA1D P25100 1/20 0.40
HTR1B P28222 1/20 0.40
HTR2C P28335 1/20 0.40
HTR1E P28566 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8449438 1.00 SIGMAR1 (0.45) SIGMAR1GRM2L3MBTL1ITGB3ITGA2B
SCHEMBL8453538 1.00 SIGMAR1 (0.45) SIGMAR1GRM2L3MBTL1ITGB3ITGA2B
SCHEMBL8948780 0.91 ITGB3 (0.51) SIGMAR1GRM2L3MBTL1ITGB3ITGA2B
SCHEMBL8455801 0.87 ITGB3 (0.54) SIGMAR1GRM2ITGB3ITGA2BHRH1
SCHEMBL8948773 0.87 SIGMAR1 (0.44) SIGMAR1GRM2L3MBTL1ITGB3ITGA2B
SCHEMBL8948876 0.85 SIGMAR1 (0.43) SIGMAR1GRM2L3MBTL1ITGB3ITGA2B
SCHEMBL8453773 0.85 GRM2 (0.51) SIGMAR1GRM2ITGB3ITGA2B
SCHEMBL8948726 0.85 GRM2 (0.52) SIGMAR1GRM2ITGB3ITGA2B
SCHEMBL8948663 0.85 L3MBTL1 (0.49) SIGMAR1GRM2L3MBTL1ITGB3ITGA2B
SCHEMBL8948589 0.85 L3MBTL1 (0.49) SIGMAR1GRM2L3MBTL1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5532255-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-07-02 US disclosed