SCHEMBL8949158

SCHEMBL8949158

COC(=O)NC(=N)c1ccc(-c2cc(C(=O)N(C)[C@H]3CC[C@H](C(=O)O)CC3)c(=O)n(C)n2)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 3/20 0.34
PDE10A Q9Y233 4/20 0.33
FASN P49327 2/20 0.32
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
VCP P55072 1/20 0.31
ROCK2 O75116 1/20 0.31
HRH3 Q9Y5N1 2/20 0.31
ALDH1A1 P00352 2/20 0.30
TYK2 P29597 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
HSD17B10 Q99714 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30
HPGD P15428 2/20 0.30
SMO Q99835 1/20 0.30
MEN1 O00255 1/20 0.30
HTT P42858 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8949191 0.88 SYK (0.36) PDE10AADORA2AADORA1ROCK2MEN1
SCHEMBL8949134 0.87 ITGB3 (0.38) PDE10AADORA2AADORA1HRH3
SCHEMBL8949140 0.87 ITGB3 (0.38) PDE10AADORA2AADORA1HRH3
SCHEMBL8949284 0.82 F2 (0.38) EGLN1PDE10AHRH3
SCHEMBL8949279 0.82 F2 (0.38) EGLN1PDE10AHRH3
Hydrochloric Acid SCHEMBL8949003 0.82 F2 (0.37) EGLN1PDE10AHRH3
SCHEMBL8949258 0.77 CNR2 (0.41) HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL8949056 0.77 CNR2 (0.41) HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL8885599 0.72 FASN (0.43) FASNROCK2ALDH1A1MEN1KMT2A
SCHEMBL8948977 0.72 FAAH (0.41) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed