SCHEMBL8949232

SCHEMBL8949232

COC(=O)C1CCC(Nc2ccc(-c3ccc(C#N)cc3)nn2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 1/20 0.43
PDGFRA P16234 1/20 0.43
KDM4E B2RXH2 1/20 0.42
CCNK O75909 4/20 0.42
CDK12 Q9NYV4 4/20 0.42
CCNA2 P20248 3/20 0.42
CDK2 P24941 3/20 0.42
CCR6 P51684 5/20 0.41
PDK1 Q15118 2/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
HPGD P15428 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NLRP3 Q96P20 1/20 0.39
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8949227 1.00 PDGFRB (0.43) PDGFRBPDGFRAKDM4ECCNKCDK12
SCHEMBL8949216 0.81 PDGFRB (0.43) PDGFRBPDGFRAPDK1PDK2PDK3
SCHEMBL8949224 0.81 PDGFRB (0.43) PDGFRBPDGFRAPDK1PDK2PDK3
SCHEMBL29817860 0.79 ACHE (0.48) PDGFRBPDGFRAPDK1HPGDRAB9A
SCHEMBL8949132 0.79 KCNH2 (0.43) KDM4ECCNKCDK12CCNA2CDK2
SCHEMBL8948987 0.75 CASP1 (0.54) KDM4ERAB9ANPC1
SCHEMBL8948991 0.75 CASP1 (0.54) KDM4ERAB9ANPC1
SCHEMBL8949241 0.74 NPC1 (0.45) KDM4ERAB9ANPC1
SCHEMBL8949251 0.74 NPC1 (0.45) KDM4ERAB9ANPC1
SCHEMBL8409339 0.73 NPC1 (0.61) RAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed