SCHEMBL8949324

SCHEMBL8949324

COC(=O)[C@H]1CC[C@H](NC(=O)c2cc(-c3ccc(C#N)cc3)nnc2N2CCOCC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 1/20 0.41
MAPK14 Q16539 2/20 0.40
CNR2 P34972 2/20 0.40
LCK P06239 1/20 0.40
KIT P10721 1/20 0.40
KDR P35968 1/20 0.40
MAPK9 P45984 1/20 0.40
TTK P33981 2/20 0.39
EGLN1 Q9GZT9 3/20 0.39
BMPR1B O00238 1/20 0.39
BMPR1A P36894 1/20 0.39
TGFBR1 P36897 1/20 0.39
ACVRL1 P37023 1/20 0.39
ACVR1 Q04771 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CFTR P13569 1/20 0.38
IRAK4 Q9NWZ3 4/20 0.38
TNF P01375 3/20 0.38
CHEK1 O14757 1/20 0.38
CD274 Q9NZQ7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8949333 1.00 HCRTR2 (0.41) HCRTR2MAPK14CNR2LCKKIT
Hydrochloric Acid SCHEMBL8949417 0.85 MAPK14 (0.42) HCRTR2MAPK14CNR2LCKKIT
SCHEMBL8948987 0.82 CASP1 (0.54) EGLN1CFTRIRAK4CHEK1
SCHEMBL8948991 0.82 CASP1 (0.54) EGLN1CFTRIRAK4CHEK1
SCHEMBL9260471 0.79 CNR2 (0.41) CNR2TTKEGLN1CFTRIRAK4
Hydrochloric Acid SCHEMBL8949020 0.77 TMPRSS15 (0.39) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL8949141 0.77 EGLN1 (0.45) CNR2TTKEGLN1CFTRIRAK4
SCHEMBL8949256 0.77 EGLN1 (0.45) CNR2TTKEGLN1CFTRIRAK4
SCHEMBL8949262 0.77 EGLN1 (0.45) CNR2TTKEGLN1CFTRIRAK4
Hydrochloric Acid SCHEMBL8949012 0.76 MAPK13 (0.40) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed