SCHEMBL8949352

SCHEMBL8949352

N=C(N)c1ccc(-c2cnc(C(=O)NCCCC(=O)O)nc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.50
ITGA2B P08514 14/20 0.50
F10 P00742 2/20 0.47
MAPK1 P28482 1/20 0.46
PPARG P37231 1/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8949087 0.96 ITGB3 (0.55) ITGB3ITGA2BF10MAPK1
Hydrochloric Acid SCHEMBL8949145 0.86 ALDH1A1 (0.46) ITGB3ITGA2BF10KDM4EALDH1A1
SCHEMBL8409855 0.86 MAPK1 (0.62) ITGB3ITGA2BF10MAPK1PPARG
Hydrochloric Acid SCHEMBL8949026 0.83 TMPRSS15 (0.45) ITGB3ITGA2BF10ALDH1A1
Hydrochloric Acid SCHEMBL8408094 0.81 MAPK1 (0.68) ITGB3ITGA2BF10MAPK1
SCHEMBL8949326 0.79 F10 (0.39) ITGB3ITGA2BF10
SCHEMBL8407980 0.77 F10 (0.60) ITGB3ITGA2BF10MAPK1CA1
SCHEMBL8948975 0.76 ITGB3 (0.50) ITGB3ITGA2B
SCHEMBL7306809 0.73 ITGB3 (0.70) ITGB3ITGA2BF10MAPK1CA1
SCHEMBL8949046 0.72 ITGB3 (0.50) ITGB3ITGA2BMAPK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed