SCHEMBL8949520

SCHEMBL8949520

COC(=O)c1ccc2oc3cc(O)ccc3c(=O)c2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.56
ALDH1A1 P00352 5/20 0.52
KDM4E B2RXH2 4/20 0.52
HPGD P15428 3/20 0.52
HSD17B10 Q99714 3/20 0.52
MEN1 O00255 1/20 0.52
TP53 P04637 1/20 0.52
CYP2C9 P11712 1/20 0.52
PTGER1 P34995 1/20 0.52
PTGER3 P43115 1/20 0.52
PTGER2 P43116 1/20 0.52
KMT2A Q03164 1/20 0.52
PTGDR Q13258 1/20 0.52
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
ESR2 Q92731 2/20 0.50
GLA P06280 2/20 0.50
GAA P10253 2/20 0.50
ESR1 P03372 1/20 0.50
KDM5A P29375 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10452782 0.95 MAOA (0.56) MAOAALDH1A1KDM4EHPGDHSD17B10
SCHEMBL11319698 0.92 KDM4E (0.56) MAOAALDH1A1KDM4EHPGDHSD17B10
SCHEMBL69937 0.89 NPC1 (0.58) MAOAALDH1A1KDM4EHPGDHSD17B10
SCHEMBL11868305 0.86 NPC1 (0.66) MAOAALDH1A1KDM4EHPGDHSD17B10
SCHEMBL11866301 0.86 THRB (0.54) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL9147000 0.86 AKR1B1 (0.58) MAOAALDH1A1KDM4EHPGDHSD17B10
SCHEMBL3966330 0.85 CREBBP (0.56) MAOAALDH1A1KDM4EHPGDHSD17B10
SCHEMBL11319692 0.85 NPC1 (0.71) MAOAALDH1A1KDM4EHPGDHSD17B10
SCHEMBL11860960 0.84 KMT2A (0.50) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL2628179 0.84 NPC1 (0.52) ALDH1A1KDM4EHPGDHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5552441-A ANTIALLERGENS, ANTIINFLAMMATORY AGENTS AND RESPIRATORY SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1996-09-03 US disclosed
EP-0442748-B1 Improvements in and relating to leukotriene antagonists LILLY CO ELI (US) 1995-01-11 EP disclosed
US-5324743-A Leukotriene B4 antagonists ELI LILLY AND COMPANY (US) 1994-06-28 US disclosed
EP-0442748-A1 Improvements in and relating to leukotriene antagonists ELI LILLY AND COMPANY (US) 1991-08-21 EP disclosed
US-4996230-A Antiallergens, antiinflammatory agent ELI LILLY AND COMPANY (US) 1991-02-26 US disclosed
US-3949084-A Novel substituted xanthone carboxylic acid compounds SYNTEX (U.S.A.) INC. (US) 1976-04-06 US disclosed