SCHEMBL8950201

SCHEMBL8950201

CN1Sc2sccc2C=C1CN1CCOCC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.43
HRH3 Q9Y5N1 3/20 0.36
CYP2A13 Q16696 4/20 0.36
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MEN1 O00255 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
CXCR4 P61073 1/20 0.35
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
KDM1A O60341 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9058336 0.80 HTT (0.36) HTTHRH3ALDH1A1KMT2ASMN1; SMN2
SCHEMBL9057846 0.76 KMT2A (0.38) HTTALDH1A1KMT2ASMN1; SMN2KDM1A
SCHEMBL9057893 0.72 CA2 (0.50) HRH3
SCHEMBL8950339 0.66 CA2 (0.41) HTTHRH3ALDH1A1KMT2ASMN1; SMN2
SCHEMBL10725828 0.64 HTT (0.53) HTTHRH3CYP2A13ALDH1A1KMT2A
SCHEMBL16182099 0.64 HTT (0.53) HTTHRH3CYP2A13ALDH1A1KMT2A
SCHEMBL5256185 0.62 HTT (0.54) HTTHRH3CYP2A13ALDH1A1KMT2A
SCHEMBL14080631 0.62 HTT (0.50) HTTHRH3CYP2A13ALDH1A1KMT2A
SCHEMBL14235132 0.62 HTT (0.50) HTTHRH3CYP2A13ALDH1A1KMT2A
SCHEMBL8950469 0.62 KMT2A (0.39) HTTHRH3ALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022099-A1 OPHTHALMIC COMPOSITIONS FOR TREATING GLAUCOMA ALCON LABORATORIES, INC. (US) 1996-07-25 WO disclosed
US-5538966-A ENZYME INHIBITORS FOR TREATMENT OF GLAUCOMA ALCON LABORATORIES, INC. (US) 1996-07-23 US disclosed
WO-1995019981-A1 THIENOTHIAZINE SULFONAMIDE DERIVATIVES PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS CARBONIC ANHYDRASE INHIBITORS ALCON LABORATORIES, INC. (US) 1995-07-27 WO disclosed