SCHEMBL8955369

SCHEMBL8955369

OCCCCCCCCOc1ccc(Cl)c(Cl)c1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
ALDH1A1 P00352 2/20 0.44
LMNA P02545 1/20 0.44
MRGPRX4 Q96LA9 1/20 0.43
GPR84 Q9NQS5 1/20 0.43
THRB P10828 2/20 0.40
THRA P10827 1/20 0.40
CNR2 P34972 2/20 0.38
MAPK1 P28482 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
LOX P28300 1/20 0.38
AOC3 Q16853 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11441977 0.98 TP53 (0.49) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL11450814 0.92 TP53 (0.50) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL10359843 0.86 CYP3A4 (0.47) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL27904038 0.84 TDP1 (0.67) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL8955424 0.84 TDP1 (0.67) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL28740947 0.81 GPR84 (0.43) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL8778565 0.81 MRGPRX4 (0.43) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL7228434 0.80 GPR84 (0.47) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL2097932 0.78 MRGPRX4 (0.45) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL8955786 0.78 ALDH1A1 (0.69) TP53CYP1A2CYP2D6TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516767-A PRODRUG AS HYPOGLYCEMIC AGENT SANDOZ LTD. (CH) 1996-05-14 US disclosed
US-5412137-A Hypoglycemic agents SANDOZ LTD. (CH) 1995-05-02 US disclosed