SCHEMBL8955402

SCHEMBL8955402

CC(N=NCCCC[C@H](N)C(=O)O)c1cccs1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 7/20 0.42
NOS1 P29475 7/20 0.42
NOS3 P29474 5/20 0.42
CYP1A2 P05177 2/20 0.42
TSHR P16473 2/20 0.42
CYP3A4 P08684 1/20 0.42
BLM P54132 1/20 0.41
POLB P06746 2/20 0.38
KMT2A Q03164 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
DDAH1 O94760 2/20 0.37
ALOX5 P09917 1/20 0.37
CYP2C19 P33261 3/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GSR P00390 1/20 0.36
GLA P06280 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14334652 0.76 POLB (0.43) POLBKMT2ATDP1ALOX5CYP2C19
SCHEMBL14335054 0.71 KIF11 (0.40) POLBKMT2ATDP1ALOX5CYP2C19
SCHEMBL8955926 0.69 HDAC1 (0.38) TSHRPOLBKMT2ATDP1ALOX5
SCHEMBL9130354 0.67 KIF11 (0.39) POLBKMT2ATDP1ALOX5CYP2C19
SCHEMBL9130364 0.67 SLC1A3 (0.40) POLBKMT2ATDP1ALOX5CYP2C19
SCHEMBL14335268 0.66 POLB (0.43) POLBKMT2ATDP1GSR
SCHEMBL15450734 0.66 NOS2 (0.58) NOS2NOS1NOS3CYP1A2TSHR
SCHEMBL19266739 0.66 NOS2 (0.58) NOS2NOS1NOS3CYP1A2TSHR
SCHEMBL9093734 0.65 HDAC1 (0.43) TSHRPOLBALOX5CYP2C19GLA
SCHEMBL9000597 0.65 HDAC1 (0.43) TSHRPOLBALOX5CYP2C19GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0707577-A4 HEME BINDING COMPOUNDS AND USE THEREOF WISCONSIN MED COLLEGE INC (US) 1996-11-06 EP disclosed
EP-0707577-A1 HEME BINDING COMPOUNDS AND USE THEREOF MEDICAL COLLEGE OF WISCONSIN RESEARCH FOUNDATION, INC. (US) 1996-04-24 EP disclosed
WO-1995001972-A1 HEME BINDING COMPOUNDS AND USE THEREOF THE MEDICAL COLLEGE OF WISCONSIN RESEARCH FOUNDATION, INC. (US) 1995-01-19 WO disclosed