SCHEMBL8957190

SCHEMBL8957190

CCCSc1ncc(C[C@H](N)C(=O)O)n1CCc1ccccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.38
DRD2 P14416 1/20 0.36
APLNR P35414 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9509859 0.91 TP53 (0.39) TP53DRD2PTGDR2ADORA3ADORA2A
SCHEMBL8957023 0.90 TP53 (0.45) TP53
SCHEMBL8957028 0.90 TP53 (0.45) TP53
SCHEMBL9507591 0.84 FNTA (0.39) TP53DRD2ADORA3ADORA2AADORA1
SCHEMBL8954114 0.81 TP53 (0.47) TP53
SCHEMBL7056477 0.81 TP53 (0.46) TP53ADORA3ADORA2AADORA1
SCHEMBL7056482 0.81 TP53 (0.46) TP53ADORA3ADORA2AADORA1
SCHEMBL9508507 0.80 TP53 (0.36) TP53DRD2PTGDR2ADORA3ADORA2A
Hydrochloric Acid SCHEMBL9530574 0.80 MAPT (0.41) TP53DRD2APLNRADORA3ADORA2A
SCHEMBL8957161 0.79 TP53 (0.40) TP53ADORA3ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536262-A4 SUBSTITUTED HISTIDINES SMITHKLINE BEECHAM CORP (US) 1996-08-14 EP disclosed
EP-0536262-A1 SUBSTITUTED HISTIDINES SMITHKLINE BEECHAM CORPORATION (US) 1993-04-14 EP disclosed