SCHEMBL9508507

SCHEMBL9508507

CCCSc1ncc(C[C@H](N=C(c2ccccc2)c2ccccc2)C(=O)OCC)n1CCc1ccccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ADORA1 P30542 2/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
DRD2 P14416 1/20 0.33
KDM5A P29375 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
KDM5B Q9UGL1 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
EPHX2 P34913 1/20 0.33
MAPT P10636 1/20 0.33
POLB P06746 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7060687 0.92 TP53 (0.42) TP53ALDH1A1HSD17B10CYP1A2CYP3A4
SCHEMBL7060686 0.92 TP53 (0.42) TP53ALDH1A1HSD17B10CYP1A2CYP3A4
SCHEMBL9508509 0.87
SCHEMBL9509859 0.84 TP53 (0.39) TP53ALDH1A1HSD17B10ADORA1ADORA3
SCHEMBL7060690 0.81
SCHEMBL8957190 0.80 TP53 (0.38) TP53ADORA1ADORA3ADORA2ADRD2
SCHEMBL8957161 0.79 TP53 (0.40) TP53ALDH1A1HSD17B10ADORA1ADORA3
SCHEMBL8954186 0.76 TP53 (0.46) TP53ALDH1A1HSD17B10ADORA1ADORA3
SCHEMBL9507591 0.76 FNTA (0.39) TP53ADORA1ADORA3ADORA2ADRD2
Hydrochloric Acid SCHEMBL9530574 0.75 MAPT (0.41) TP53ALDH1A1HSD17B10ADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0561878-A1 USE OF ANGIOTENSIN II ANTAGONIST IN THE TREATMENT OF INFARCTION SMITHKLINE BEECHAM PLC (GB) 1993-09-29 EP disclosed