SCHEMBL8957161

SCHEMBL8957161

CCCSc1ncc(C[C@H](NC(=O)CCC)C(=O)OCC)n1CCc1ccccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.40
ADORA1 P30542 2/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ALDH1A1 P00352 4/20 0.37
MAPT P10636 3/20 0.37
LMNA P02545 1/20 0.37
THRB P10828 1/20 0.37
HSD17B10 Q99714 1/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7056937 0.92 TP53 (0.46) TP53ADORA1ADORA3ADORA2AALDH1A1
SCHEMBL9507591 0.92 FNTA (0.39) TP53ADORA1ADORA3ADORA2AMAPT
SCHEMBL8957164 0.87 TP53 (0.40) TP53ALDH1A1MAPTLMNATHRB
SCHEMBL9509859 0.84 TP53 (0.39) TP53ADORA1ADORA3ADORA2AALDH1A1
SCHEMBL7056869 0.83 TP53 (0.45) TP53ALDH1A1MAPT
SCHEMBL7056939 0.81 PTGES (0.41)
SCHEMBL9508507 0.79 TP53 (0.36) TP53ADORA1ADORA3ADORA2AALDH1A1
SCHEMBL8957190 0.79 TP53 (0.38) TP53ADORA1ADORA3ADORA2A
Hydrochloric Acid SCHEMBL9530574 0.78 MAPT (0.41) TP53ADORA1ADORA3ADORA2AALDH1A1
SCHEMBL8971303 0.77 TP53 (0.44) TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536262-A4 SUBSTITUTED HISTIDINES SMITHKLINE BEECHAM CORP (US) 1996-08-14 EP disclosed
EP-0561876-A1 USE OF ANGIOTENSIN II RECEPTOR ANTAGONISTS IN THE TREATMENT OF ATHEROMA. SMITHKLINE BEECHAM PLC (GB) 1993-09-29 EP disclosed
EP-0561901-A1 USE OF ANGIOTENSIN II RECEPTOR ANTAGONISTS IN THE TREATMENT OF DIABETIC RETINOPATHY SMITHKLINE BEECHAM PLC (GB) 1993-09-29 EP disclosed
EP-0536262-A1 SUBSTITUTED HISTIDINES SMITHKLINE BEECHAM CORPORATION (US) 1993-04-14 EP disclosed