SCHEMBL8957912

SCHEMBL8957912

Cc1cc(NC(=O)N(C)c2ccccc2)cc(C)c1S(=O)(=O)C[N+](=O)[O-]

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 2/20 0.43
ATM Q13315 1/20 0.38
MLYCD O95822 1/20 0.38
IMPDH2 P12268 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
THRA P10827 2/20 0.37
THRB P10828 1/20 0.37
SENP1 Q9P0U3 2/20 0.37
AKR1B1 P15121 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8957970 0.84 CA12 (0.41)
SCHEMBL8957976 0.83 LMNA (0.48) NPC1RAB9ASMN1; SMN2KDM4EMEN1
SCHEMBL8958053 0.80 CA12 (0.40) SMN1; SMN2KDM4EATMMEN1KMT2A
SCHEMBL8467038 0.79 ALDH1A1 (0.52) SMN1; SMN2MEN1KMT2AAKR1B1
SCHEMBL7223994 0.79 POLB (0.36) RAB9AKDM4EMEN1KMT2AAKR1B1
SCHEMBL7228473 0.79 MAPT (0.40) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL8958001 0.78 CA12 (0.40) NPC1RAB9AMEN1KMT2ATHRB
SCHEMBL8957820 0.78 THRA (0.38) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL7223364 0.78 POLB (0.45) NPC1RAB9AMEN1KMT2AAKR1B1
SCHEMBL7225299 0.78 ALDH1A1 (0.43) SMN1; SMN2KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0469889-B1 (p-Carbonylaminophenyl)-sulphonyl-nitromethane derivatives ZENECA LTD (GB) 1996-01-17 EP disclosed
US-5189031-A Inhibitor of enzyme aldose reductase, useful in the treatment of certain peripheral effects of diabetes and galactosemia IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-02-23 US disclosed
US-5110808-A Aldose reductase inhibitors; peripheral effects of diabetes and galactosemia IMPERIAL CHEMICAL INDUSTRIES, PLC (GB) 1992-05-05 US disclosed
EP-0469889-A1 (p-Carbonylaminophenyl)-sulphonyl-nitromethane derivatives ZENECA LIMITED (GB) 1992-02-05 EP disclosed