SCHEMBL8957970

SCHEMBL8957970

Cc1cc(NC(=O)N(C)C)cc(C)c1S(=O)(=O)C[N+](=O)[O-]

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH1A1 P00352 1/20 0.39
APEX1 P27695 1/20 0.36
TSHR P16473 1/20 0.36
GAA P10253 1/20 0.35
PTGES O14684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9592058 0.87 ALDH1A1 (0.32) ALDH1A1GAA
SCHEMBL8958053 0.87 CA12 (0.40) CA12CA1CA2CA9ALDH1A1
SCHEMBL7223994 0.86 POLB (0.36) ALDH1A1GAA
SCHEMBL7228473 0.86 MAPT (0.40) CA12CA1CA2CA9ALDH1A1
SCHEMBL7225299 0.85 ALDH1A1 (0.43) ALDH1A1GAA
SCHEMBL7223364 0.85 POLB (0.45) ALDH1A1GAA
SCHEMBL8957912 0.84 NPC1 (0.43)
SCHEMBL8957992 0.84 KMT2A (0.51) CA12CA1CA2CA9ALDH1A1
SCHEMBL7230766 0.83 POLB (0.42) ALDH1A1GAA
SCHEMBL8958259 0.83 RAB9A (0.34) ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0469889-B1 (p-Carbonylaminophenyl)-sulphonyl-nitromethane derivatives ZENECA LTD (GB) 1996-01-17 EP disclosed
US-5189031-A Inhibitor of enzyme aldose reductase, useful in the treatment of certain peripheral effects of diabetes and galactosemia IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-02-23 US disclosed
US-5110808-A Aldose reductase inhibitors; peripheral effects of diabetes and galactosemia IMPERIAL CHEMICAL INDUSTRIES, PLC (GB) 1992-05-05 US disclosed
EP-0469889-A1 (p-Carbonylaminophenyl)-sulphonyl-nitromethane derivatives ZENECA LIMITED (GB) 1992-02-05 EP disclosed