SCHEMBL8959155

SCHEMBL8959155

CCOC(=O)c1cc2ccc(N)cc2[nH]1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.70
KDM4E B2RXH2 4/20 0.63
ALDH1A1 P00352 4/20 0.63
HPGD P15428 3/20 0.63
RAB9A P51151 3/20 0.63
LMNA P02545 3/20 0.63
SMN1; SMN2 Q16637 2/20 0.63
NPC1 O15118 2/20 0.63
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
GLA P06280 1/20 0.63
GAA P10253 1/20 0.63
MAPT P10636 1/20 0.63
ATM Q13315 1/20 0.63
HSD17B10 Q99714 2/20 0.61
MMP13 P45452 8/20 0.59
MMP2 P08253 6/20 0.59
HTT P42858 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
HRH3 Q9Y5N1 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL656018 0.88 KDM4E (0.74) ALOX15KDM4EALDH1A1HPGDRAB9A
Hydrochloric Acid SCHEMBL28674698 0.87 KDM4E (0.72) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL5623372 0.85 KDM4E (0.78) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL17368519 0.84 ALOX15 (0.72) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL71101 0.84 ALOX15 (0.72) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL4907791 0.84 ALOX15 (0.72) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL654862 0.83 HRH4 (0.55) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL17092514 0.83 HRH4 (0.55) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL327597 0.83 MMP13 (0.80) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL5917481 0.82 ALOX15 (0.70) ALOX15KDM4EALDH1A1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0424261-B1 Dyeing composition containing oxidation dyes precursors and aminoindole derivatives as coupling agent OREAL (FR) 1996-01-03 EP claimed
EP-0425345-B1 Keratinic fibres dyeing process with amino-indoles, composition and use devices OREAL (FR) 1994-09-14 EP claimed
EP-0460996-B1 Keratinic fibres dyeing process with an aminoindol associated with a quinone derivative OREAL (FR) 1994-09-14 EP claimed
US-5254135-A Applying indole dye, developing with oxidizing system L'OREAL (FR) 1993-10-19 US claimed
US-5180400-A METHOD FOR DYEING KERATINOUS FIBRES USING AN AMINOINDOLE IN COMBINATION WITH A QUINONE DERIVATIVE L'OREAL (FR) 1993-01-19 US claimed
EP-0460996-A1 Keratinic fibres dyeing process with an aminoindol associated with a quinone derivative L'OREAL (FR) 1991-12-11 EP claimed
EP-0425345-A1 Keratinic fibres dyeing process with amino-indoles, composition and use devices L'OREAL (FR) 1991-05-02 EP claimed
EP-0424261-A1 Dyeing composition containing oxidation dyes precursors and aminoindole derivatives as coupling agent L'OREAL (FR) 1991-04-24 EP claimed
EP-3882245-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2021-09-22 EP disclosed
CN-111808079-A Indole ASK1 small molecule inhibitor and preparation method and application thereof 中国药科大学 2020-10-23 CN disclosed
CN-108191858-B A kind of intermediate preparing pyrroloquinoline quinone and preparation method 山东康迈祺生物科技有限公司 2019-11-26 CN disclosed
US-10183932-B2 Substituted oxopyridine derivatives and use thereof cardiovascular disorders BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-01-22 US disclosed
CN-108191858-A A kind of intermediate and preparation method for preparing pyrroloquinoline quinone 山东康迈祺生物科技有限公司 2018-06-22 CN disclosed
CN-107089982-B 4, 5-disubstituted-1-hydrogen-pyrrole (2, 3-f) quinoline-2, 7, 9-tricarboxylate compound and application thereof 王靖林 2018-06-05 CN disclosed
EP-0602851-A1 Quinazoline derivatives ZENECA LIMITED (GB) 1994-06-22 EP disclosed
US-5254135-A Applying indole dye, developing with oxidizing system L'OREAL (FR) 1993-10-19 US disclosed
US-5180400-A METHOD FOR DYEING KERATINOUS FIBRES USING AN AMINOINDOLE IN COMBINATION WITH A QUINONE DERIVATIVE L'OREAL (FR) 1993-01-19 US disclosed
EP-0460996-A1 Keratinic fibres dyeing process with an aminoindol associated with a quinone derivative L'OREAL (FR) 1991-12-11 EP disclosed
EP-0425345-A1 Keratinic fibres dyeing process with amino-indoles, composition and use devices L'OREAL (FR) 1991-05-02 EP disclosed
EP-0424261-A1 Dyeing composition containing oxidation dyes precursors and aminoindole derivatives as coupling agent L'OREAL (FR) 1991-04-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10183932-B2 Substituted oxopyridine derivatives and use thereof cardiovascular disorders OGFOD1, VASP, PNPO ALOX15 608/4885KDM4E 1342/4885ALDH1A1 1195/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.