SCHEMBL8959454

SCHEMBL8959454

CC(CN1CC(=O)N(C)c2ccc(I)cc2C1=O)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.44
ITGB3 P05106 3/20 0.42
ITGA2B P08514 3/20 0.42
PRMT5 O14744 1/20 0.42
WDR77 Q9BQA1 1/20 0.42
MDM2 Q00987 7/20 0.41
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRA6 Q16445 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
TP53 P04637 1/20 0.35
DNMT1 P26358 1/20 0.34
MAPT P10636 2/20 0.34
HPGD P15428 2/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7329048 0.88 CASP3 (0.41) CASP3ITGB3ITGA2BPRMT5WDR77
SCHEMBL7325381 0.75 ITGB3 (0.46) CASP3ITGB3ITGA2BGABRA1GABRG2
Trifluoroacetic Acid SCHEMBL7323917 0.75 ITGB3 (0.37) ITGB3ITGA2BPRMT5WDR77GABRA1
SCHEMBL7357974 0.74 ITGB3 (0.50) ITGB3ITGA2B
SCHEMBL7329841 0.73 ITGB3 (0.44) CASP3ITGB3ITGA2BPRMT5WDR77
SCHEMBL7319919 0.70 ITGB3 (0.48) CASP3ITGB3ITGA2BMDM2GABRA1
SCHEMBL2833423 0.68 CASP3 (0.51) CASP3MAPTALDH1A1
SCHEMBL7322279 0.67 MEN1 (0.40) CASP3ITGB3ITGA2BMDM2TP53
SCHEMBL1500258 0.67 SDCBP (0.52) PRMT5WDR77DPP7DNMT1KDM4E
SCHEMBL8959460 0.67 KDM4E (0.47) ITGB3ITGA2BMDM2TP53DNMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0610334-B1 NONPEPTIDYL INTEGRIN INHIBITORS HAVING SPECIFICITY FOR THE GPII B III A RECEPTOR GENENTECH INC (US) 1996-01-24 EP disclosed