SCHEMBL8959486

SCHEMBL8959486

NC(Cn1ccc2cc(Cl)ccc21)OC(=O)/C=C/C(=O)OC(N)Cn1ccc2cc(Cl)ccc21

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.58
HTR2A P28223 7/20 0.58
PRMT5 O14744 1/20 0.42
KRAS P01116 2/20 0.40
ACLY P53396 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
OXER1 Q8TDS5 1/20 0.39
KMO O15229 1/20 0.39
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
HTR2B P41595 1/20 0.37
NPY5R Q15761 1/20 0.36
CDK4 P11802 1/20 0.36
CCND1 P24385 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7673292 0.90 KMO (0.50) HTR2CHTR2APRMT5ACLYOXER1
SCHEMBL8959694 0.85 HTR2C (0.58) HTR2CHTR2APRMT5HDAC3HDAC1
SCHEMBL8959627 0.82 HTR2C (0.60) HTR2CHTR2AKRASHDAC1HDAC8
SCHEMBL8959507 0.78 HTR2C (0.60) HTR2CHTR2AKRASCYP1A2CYP3A4
SCHEMBL4042963 0.78 HTR2C (0.65) HTR2CHTR2APRMT5ACLYHDAC3
SCHEMBL4042962 0.78 HTR2C (0.65) HTR2CHTR2APRMT5ACLYHDAC3
Fumaric Acid SCHEMBL7091385 0.78 HTR2C (0.78) HTR2CHTR2APRMT5KRASACLY
Fumaric Acid SCHEMBL7091387 0.78 HTR2C (0.78) HTR2CHTR2APRMT5KRASACLY
SCHEMBL7677260 0.78 HTR2C (0.45) HTR2CHTR2APRMT5HDAC3HDAC1
SCHEMBL3951044 0.76 HTR2C (0.63) HTR2CHTR2APRMT5KRASACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed