SCHEMBL8959541

SCHEMBL8959541

CCc1c(C(=O)O)[nH]c2ccc(F)cc12

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRNP P04156 1/20 0.69
CYP1A2 P05177 1/20 0.69
CYP2C9 P11712 1/20 0.69
CYP2C19 P33261 1/20 0.69
PPARG P37231 1/20 0.69
HIF1A Q16665 1/20 0.69
NPSR1 Q6W5P4 1/20 0.69
RXFP1 Q9HBX9 1/20 0.69
NR2E3 Q9Y5X4 1/20 0.69
NCOR2 Q9Y618 1/20 0.69
KDM4E B2RXH2 3/20 0.56
CNR1 P21554 4/20 0.55
PTGS1 P23219 1/20 0.49
PTGS2 P35354 1/20 0.49
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
HSD17B10 Q99714 1/20 0.48
MAP2 P11137 1/20 0.48
GPR17 Q13304 1/20 0.47
DRD2 P14416 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7411140 0.85 KDM4E (0.71) PRNPCYP1A2CYP2C9CYP2C19PPARG
SCHEMBL1553071 0.83 NPSR1 (0.71) PRNPCYP1A2CYP2C9CYP2C19PPARG
SCHEMBL3107611 0.83 PRNP (0.71) PRNPCYP1A2CYP2C9CYP2C19PPARG
SCHEMBL8959676 0.83 DRD2 (0.62) PRNPCYP1A2CYP2C9CYP2C19PPARG
SCHEMBL1894184 0.82 RXFP1 (1.00) PRNPCYP1A2CYP2C9CYP2C19PPARG
SCHEMBL2538695 0.82 PRNP (0.69) PRNPCYP1A2CYP2C9CYP2C19PPARG
SCHEMBL2730323 0.81 ALDH1A1 (0.59) CYP2C19KDM4ECNR1PTGS1PTGS2
SCHEMBL3036074 0.79 KDM4E (0.74) PRNPCYP1A2CYP2C9CYP2C19PPARG
SCHEMBL24196991 0.79 CNR1 (0.52) PRNPCYP1A2CYP2C9CYP2C19PPARG
SCHEMBL9231630 0.78 DRD2 (0.44) PRNPCYP1A2CYP2C9CYP2C19PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
CN-1105988-A 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 CN disclosed
EP-0655440-A2 1-Aminoethylindoles F. HOFFMANN-LA ROCHE AG (CH) 1995-05-31 EP disclosed