SCHEMBL8959984

SCHEMBL8959984

COc1c[nH]c2cccc(C)c12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.55
HTR2A P28223 6/20 0.49
HTR2B P41595 2/20 0.46
HTR6 P50406 1/20 0.46
HTR2C P28335 1/20 0.46
HTR1A P08908 1/20 0.41
HTR7 P34969 1/20 0.41
HTR5A P47898 1/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
MMP9 P14780 1/20 0.40
ATM Q13315 2/20 0.39
NR4A2 P43354 1/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
IDO1 P14902 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL788913 0.85 HTR2A (0.57) GPR84HTR2AHTR2BHTR6HTR2C
SCHEMBL28167758 0.84 HTR2A (0.60) HTR2AHTR2BHTR6HTR2CHTR1A
SCHEMBL31744662 0.81 GPR84 (0.44) GPR84HTR2AHTR6KDM4EMAPT
SCHEMBL28167759 0.79 FFAR1 (0.53) GPR84HTR2AHTR2BHTR6HTR2C
SCHEMBL28337297 0.79 NR4A2 (0.55) GPR84HTR2AHTR2BHTR6HTR2C
SCHEMBL30089577 0.79 HTR2A (0.50) HTR2AHTR2BHTR6HTR2CHTR1A
SCHEMBL27920584 0.78 SLC22A6 (0.59) GPR84HTR2AMTNR1AMTNR1BNR4A2
SCHEMBL1224614 0.77 GPR84 (0.64) GPR84HTR2AHTR2BHTR2CATM
SCHEMBL30552280 0.77 GPR84 (0.64) GPR84HTR2AHTR2BHTR2CATM
SCHEMBL27772015 0.74 GPR84 (0.44) GPR84HTR2AMTNR1AMTNR1BNR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
EP-0655440-A2 1-Aminoethylindoles F. HOFFMANN-LA ROCHE AG (CH) 1995-05-31 EP disclosed