SCHEMBL8960071

SCHEMBL8960071

COc1ccc(C2=CCCNC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.56
ADRA2B P18089 1/20 0.56
HTR2A P28223 3/20 0.52
HTR2C P28335 1/20 0.52
HTR2B P41595 1/20 0.52
HTR6 P50406 1/20 0.46
NISCH Q9Y2I1 1/20 0.41
KCNH2 Q12809 1/20 0.41
RYR2 Q92736 1/20 0.41
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
ADRB1 P08588 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14085315 0.81 QDPR (0.43) HTR2CHTR6NISCHSIGMAR1CA12
SCHEMBL11195019 0.80 HTR2A (0.51) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL8960144 0.79 ADRA2A (0.61) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL29140058 0.79 ADRA2A (0.53) ADRA2AADRA2BHTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL11191756 0.79 HTR2A (0.50) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL11198805 0.78 ADRA2A (0.55) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL169373 0.76 HTR2A (0.50) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL8960083 0.76 ADRA2A (0.61) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL29140051 0.76 ADRA2A (0.61) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL8960049 0.76 ADRA2A (0.61) ADRA2AADRA2BHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109810047-A (R) synthetic method of the chiral intermediate of -3- Phenylpiperidine or/and (S) -3- Phenylpiperidine and Ni Lapani 上海博邦医药科技有限公司 2019-05-28 CN disclosed
EP-0691956-A1 3-PHENYL-1,2,5,6-TETRAHYDROPYRIDINE DERIVATIVES AS SEDATIVES LABORATOIRE L. LAFON (FR) 1996-01-17 EP disclosed
WO-1994022827-A1 3-PHENYL-1,2,5,6-TETRAHYDROPYRIDINE DERIVATIVES AS SEDATIVES LABORATOIRE L. LAFON (FR) 1994-10-13 WO disclosed