SCHEMBL8961445

SCHEMBL8961445

NCCNC(=O)CN1CCCC1=O

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.57
HTT P42858 1/20 0.54
KMT2A Q03164 4/20 0.48
NQO2 P16083 1/20 0.46
LMNA P02545 1/20 0.45
ADRA1D P25100 4/20 0.42
ADRA1A P35348 4/20 0.42
ADRA1B P35368 4/20 0.42
ATAD2 Q6PL18 1/20 0.41
CECR2 Q9BXF3 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
MAPK1 P28482 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11242670 0.90 HTT (0.59) TSHRHTTKMT2ANQO2LMNA
SCHEMBL9208885 0.85 HTT (0.55) TSHRHTTKMT2ANQO2LMNA
SCHEMBL11245716 0.85 HTT (0.55) TSHRHTTKMT2ANQO2LMNA
SCHEMBL5255092 0.83 HTT (0.52) TSHRHTTKMT2ANQO2LMNA
SCHEMBL9851181 0.83 KMT2A (0.58) TSHRKMT2ASMN1; SMN2MAPK1ALDH1A1
SCHEMBL9628927 0.81 TSHR (0.67) TSHRHTTKMT2ANQO2LMNA
SCHEMBL11384074 0.81 HTT (0.50) TSHRHTTKMT2ANQO2LMNA
SCHEMBL11553497 0.80 HTT (0.50) TSHRHTTKMT2ANQO2LMNA
SCHEMBL20618032 0.80 LMNA (0.51) TSHRHTTKMT2ANQO2LMNA
SCHEMBL8961486 0.80 LMNA (0.51) TSHRHTTKMT2ANQO2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299495-B1 1-Pyrrolidineacetamide derivatives and use thereof SANWA KAGAKU KENKYUSHO CO (JP) 1996-02-07 EP disclosed
EP-0408524-B1 (Pyrrolidin-2-on-l-yl) acetamides as enhancers of learning and memory and pharmaceutical compositions comprising same SIGMA TAU IND FARMACEUTI (IT) 1995-11-08 EP disclosed
US-5061725-A COGNITION ACTIVATORS SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 1991-10-29 US disclosed
EP-0408524-A1 (Pyrrolidin-2-on-l-yl) acetamides as enhancers of learning and memory and pharmaceutical compositions comprising same Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 1991-01-16 EP disclosed
US-4939126-A 1-pyrrolidineacetamide derivatives and use thereof SANWA KAGAKU KENKYUSHO CO. LTD. (JP) 1990-07-03 US disclosed
EP-0299495-A2 1-Pyrrolidineacetamide derivatives and use thereof SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1989-01-18 EP disclosed