SCHEMBL8964600

SCHEMBL8964600

C=CCc1ccc(OC)cc1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
TP53 P04637 1/20 0.53
CYP3A4 P08684 1/20 0.53
ALOX15 P16050 1/20 0.53
TSHR P16473 1/20 0.53
ALOX12 P18054 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
FFAR4 Q5NUL3 1/20 0.46
MAPT P10636 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SLC2A1 P11166 1/20 0.41
PPARG P37231 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41
APLNR P35414 1/20 0.41
PTPN1 P18031 2/20 0.40
KDM1A O60341 1/20 0.40
MAOA P21397 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2096402 0.85 ALDH1A1 (0.57) ALDH1A1TP53CYP3A4ALOX15TSHR
SCHEMBL22700982 0.82 ALDH1A1 (0.48) ALDH1A1TP53CYP3A4ALOX15TSHR
SCHEMBL10725515 0.82 NQO1 (0.43) ALDH1A1TP53CYP3A4ALOX15TSHR
SCHEMBL2559819 0.81 HTT (0.45) ALDH1A1APLNRKDM1AMAOAMAOB
SCHEMBL30105464 0.81 APLNR (0.58) ALDH1A1TP53CYP3A4ALOX15TSHR
SCHEMBL2845262 0.81 APLNR (0.58) ALDH1A1TP53CYP3A4ALOX15TSHR
SCHEMBL2843664 0.80 PTPN1 (0.54) ALDH1A1TP53CYP3A4ALOX15TSHR
SCHEMBL12717376 0.80 ALDH1A1 (0.52) ALDH1A1TP53CYP3A4ALOX15TSHR
SCHEMBL14775356 0.80 L3MBTL1 (0.38) ALDH1A1TP53CYP3A4ALOX15TSHR
SCHEMBL9226953 0.79 ALDH1A1 (0.50) ALDH1A1TP53CYP3A4ALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0410379-B1 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMA (US) 1996-01-31 EP disclosed
US-5068465-A Hypotensive agents or enzyme inhibitors for treatment of hypertension MERRELL DOW PHARMACEUTICALS INC. (US) 1991-11-26 US disclosed
EP-0410379-A2 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMACEUTICALS INC. (US) 1991-01-30 EP disclosed
US-4981868-A ENZYME INHIBITORS, HYPOTENSIVES MERRELL DOW PHARMACEUTICAL (US) 1991-01-01 US disclosed