SCHEMBL8965432

SCHEMBL8965432

COc1cccc(C(Cc2ccccc2)C(=O)OC(C)(C)C)c1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 4/20 0.54
MTNR1B P49286 4/20 0.54
ITGA4 P13612 1/20 0.46
ITGB7 P26010 1/20 0.46
CASR P41180 1/20 0.46
GPR139 Q6DWJ6 1/20 0.46
CHRM1 P11229 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
POLB P06746 1/20 0.43
RAB9A P51151 1/20 0.43
KDM4E B2RXH2 1/20 0.43
BCHE P06276 1/20 0.43
USP2 O75604 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7042372 0.87 MTNR1A (0.62) MTNR1AMTNR1BCASRGPR139CHRM1
SCHEMBL7041441 0.84 MTNR1A (0.61) MTNR1AMTNR1BCASRGPR139L3MBTL1
SCHEMBL21656313 0.83 L3MBTL1 (0.50) MTNR1AMTNR1BCHRM1L3MBTL1KDM4E
SCHEMBL27555215 0.83 MTNR1A (0.63) MTNR1AMTNR1BCASRGPR139L3MBTL1
SCHEMBL28617579 0.82 EPHX1 (0.65) MTNR1AMTNR1BCASRGPR139L3MBTL1
SCHEMBL8912764 0.82 MTNR1A (0.58) MTNR1AMTNR1BCASRGPR139L3MBTL1
SCHEMBL29609868 0.82 EPHX1 (0.65) MTNR1AMTNR1BCASRGPR139L3MBTL1
SCHEMBL4239829 0.81 ITGA4 (0.47) ITGA4ITGB7POLBRAB9AKDM4E
SCHEMBL10202970 0.79 MTNR1A (0.55) MTNR1AMTNR1BCASRCHRM1POLB
SCHEMBL30854869 0.77 KMT2A (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0593557-B1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME (GB) 1996-01-31 EP disclosed
EP-0593557-A1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY. MERCK SHARP & DOHME (GB) 1994-04-27 EP disclosed
WO-1993001160-A1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-01-21 WO disclosed
EP-0522808-A2 Aromatic compounds, pharmaceutical compositions containing them and their use in therapy MERCK SHARP & DOHME LTD. (GB) 1993-01-13 EP disclosed