SCHEMBL8966742

SCHEMBL8966742

CCCCCCCCNCCCSc1ccncc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.45
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 2/20 0.43
PKM P14618 2/20 0.43
TSHR P16473 1/20 0.42
DRD2 P14416 2/20 0.40
DRD4 P21917 2/20 0.40
DRD3 P35462 2/20 0.40
RYR2 Q92736 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C19 P33261 2/20 0.39
MAPT P10636 1/20 0.39
HRH4 Q9H3N8 2/20 0.38
HRH3 Q9Y5N1 2/20 0.38
FDPS P14324 1/20 0.38
LMNA P02545 1/20 0.37
GPR84 Q9NQS5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8967318 1.00 NAAA (0.45) NAAAKDM4EALDH1A1PKMTSHR
SCHEMBL8966315 0.97 KDM4E (0.47) NAAAKDM4EALDH1A1PKMTSHR
SCHEMBL8966693 0.97 KDM4E (0.47) NAAAKDM4EALDH1A1PKMTSHR
SCHEMBL8966863 0.97 KDM4E (0.47) NAAAKDM4EALDH1A1PKMTSHR
SCHEMBL8966695 0.94 NAAA (0.45) NAAAKDM4EALDH1A1PKMTSHR
4-Mercaptopyridine SCHEMBL9462769 0.87 NAAA (0.40) NAAAKDM4EALDH1A1PKMTSHR
SCHEMBL9742985 0.86 GPR84 (0.46) NAAAKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL9743357 0.86 GPR84 (0.46) NAAAKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL424824 0.82 MAOA (0.49) KDM4EALDH1A1PKMCYP1A2CYP3A4
SCHEMBL8656049 0.82 CHRM2 (0.48) ALDH1A1DRD2DRD4DRD3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5561147-A ANTIINFLAMMATORY AGENT, ANTIPYRETIC, ANALGESICS, ANTIALLERGENS, IMMUNOSUPPRESSANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-01 US disclosed
US-5457106-A Antiinflammatory agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-10 US disclosed
US-5389658-A Administering as antipyretic, antiinflammatory, analgesic, antiallergic, or immunosupressive agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0612729-A2 Pyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1994-08-31 EP disclosed
US-5246948-A Antiinflammatory, antipyretic, analgesic, antiallergic, immunosupressing or immunomodulating activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-21 US disclosed
EP-0522606-A2 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-13 EP disclosed