SCHEMBL8967046

SCHEMBL8967046

COc1c(C(=O)O)cc(SC)c2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.48
KDM4E B2RXH2 6/20 0.47
ALDH1A1 P00352 5/20 0.47
HPGD P15428 5/20 0.47
NPSR1 Q6W5P4 2/20 0.47
CDC25B P30305 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
MAPK1 P28482 1/20 0.42
MCL1 Q07820 1/20 0.42
CYP1A1 P04798 1/20 0.42
CYP1B1 Q16678 1/20 0.42
HSD17B10 Q99714 2/20 0.41
ALOX15 P16050 1/20 0.41
PDE10A Q9Y233 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
IDO1 P14902 1/20 0.40
NR4A1 P22736 1/20 0.40
NR4A2 P43354 1/20 0.40
NR4A3 Q92570 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL669832 0.79 THRB (0.61) POLBKDM4EALDH1A1HPGDNPSR1
SCHEMBL976330 0.79 KDM4E (0.57) POLBKDM4EALDH1A1HPGDNPSR1
SCHEMBL8967049 0.78 ALDH1A1 (0.60) KDM4EALDH1A1HPGDNPSR1CDC25B
SCHEMBL6987407 0.78 HSD17B10 (0.56) KDM4EALDH1A1HPGDMCL1HSD17B10
SCHEMBL485446 0.78 KDM4E (0.47) KDM4EALDH1A1HPGDNPSR1CDC25B
SCHEMBL10584881 0.76 KDM4E (0.77) POLBKDM4EALDH1A1HPGDNPSR1
SCHEMBL9978740 0.75 MCL1 (0.60) KDM4EALDH1A1HPGDNPSR1CDC25B
SCHEMBL7443511 0.74 DRD3 (0.54) KDM4EALDH1A1HPGDNPSR1CDC25B
SCHEMBL1671110 0.73 CYP1A1 (0.64) KDM4EALDH1A1HPGDNPSR1CDC25B
SCHEMBL7537612 0.73 POLB (0.48) POLBKDM4EALDH1A1HPGDCDC25B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0585116-B1 1-Alkoxy-naphthalene-2-carboxamide derivatives with high affinity for the serotonin 5-HT1A receptor LILLY INDUSTRIES LTD (GB) 1996-02-28 EP disclosed
US-5389684-A Treats disorder of central nervous system LILLY INDUSTRIES LIMITED (GB) 1995-02-14 US disclosed
EP-0585116-A1 1-Alkoxy-naphthalene-2-carboxamide derivatives with high affinity for the serotonin 5-HT1A receptor LILLY INDUSTRIES LIMITED (GB) 1994-03-02 EP disclosed