SCHEMBL8967049

SCHEMBL8967049

COc1c(C(=O)O)cc(Cl)c2ccccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.60
KDM4E B2RXH2 7/20 0.60
HPGD P15428 4/20 0.60
HSD17B10 Q99714 3/20 0.60
MEN1 O00255 2/20 0.60
HTT P42858 2/20 0.60
KMT2A Q03164 2/20 0.60
MAPT P10636 1/20 0.60
PKM P14618 1/20 0.60
DRD3 P35462 2/20 0.51
DRD2 P14416 1/20 0.51
LMNA P02545 1/20 0.49
SLC2A1 P11166 1/20 0.46
CDC25B P30305 1/20 0.46
NPSR1 Q6W5P4 1/20 0.45
MAPK1 P28482 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
APEX1 P27695 1/20 0.45
NOTUM Q6P988 1/20 0.45
MCL1 Q07820 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10391302 0.87 ALDH1A1 (0.52) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL9108463 0.87 DRD3 (0.48) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL976330 0.81 KDM4E (0.57) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL669832 0.81 THRB (0.61) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL6987407 0.80 HSD17B10 (0.56) ALDH1A1KDM4EHPGDHSD17B10DRD3
SCHEMBL485446 0.80 KDM4E (0.47) ALDH1A1KDM4EHPGDHSD17B10CDC25B
SCHEMBL23725371 0.79 HIF1A (0.48) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL9110910 0.78 MCL1 (0.54) ALDH1A1KDM4EHPGDHSD17B10CDC25B
SCHEMBL8967046 0.78 POLB (0.48) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL9978740 0.78 MCL1 (0.60) ALDH1A1KDM4EHPGDHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0585116-B1 1-Alkoxy-naphthalene-2-carboxamide derivatives with high affinity for the serotonin 5-HT1A receptor LILLY INDUSTRIES LTD (GB) 1996-02-28 EP disclosed
US-5389684-A Treats disorder of central nervous system LILLY INDUSTRIES LIMITED (GB) 1995-02-14 US disclosed
EP-0585116-A1 1-Alkoxy-naphthalene-2-carboxamide derivatives with high affinity for the serotonin 5-HT1A receptor LILLY INDUSTRIES LIMITED (GB) 1994-03-02 EP disclosed