SCHEMBL8968209

SCHEMBL8968209

CC(C)(C)c1ccc(C#N)cc1NC(=NC#N)Oc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.36
CXCR2 P25025 3/20 0.35
CXCR1 P25024 2/20 0.35
LPAR1 Q92633 1/20 0.33
F2 P00734 1/20 0.33
PLG P00747 1/20 0.33
PLAU P00749 1/20 0.33
KLKB1 P03952 1/20 0.33
PRSS1 P07477 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP2C19 P33261 2/20 0.32
TRPM4 Q8TD43 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
ACP1 P24666 1/20 0.31
SLC22A12 Q96S37 1/20 0.31
ALDH1A1 P00352 3/20 0.31
USP2 O75604 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9235204 1.00 KMT2A (0.36) KMT2ACXCR2CXCR1LPAR1F2
SCHEMBL8968189 0.82 ALDH1A1 (0.43) KMT2ACXCR2CXCR1LPAR1F2
SCHEMBL8968827 0.79 CXCR2 (0.44) KMT2ACXCR2CXCR1F2PLG
SCHEMBL8968824 0.79 CXCR2 (0.44) KMT2ACXCR2CXCR1F2PLG
SCHEMBL4996687 0.76 KMT2A (0.44) KMT2AF2PLGPLAUKLKB1
SCHEMBL4996691 0.76 KMT2A (0.44) KMT2AF2PLGPLAUKLKB1
SCHEMBL5005229 0.75 ALDH1A1 (0.54) KMT2ACYP1A2CYP2C19ALDH1A1USP2
SCHEMBL14257551 0.75 ALDH1A1 (0.54) KMT2ACYP1A2CYP2C19ALDH1A1USP2
SCHEMBL5005228 0.75 ALDH1A1 (0.54) KMT2ACYP1A2CYP2C19ALDH1A1USP2
SCHEMBL14257564 0.73 RAB9A (0.43) KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547966-A Aryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1996-08-20 US disclosed
EP-0656350-A1 Biaryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1995-06-07 EP disclosed