SCHEMBL8968295

SCHEMBL8968295

COc1cc2c(c(OC)c1)N=C1CCCCCN1C2

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 13/20 0.47
HRH3 Q9Y5N1 1/20 0.41
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
BCHE P06276 2/20 0.38
ALDH1A1 P00352 2/20 0.37
LMNA P02545 2/20 0.37
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37
CYP3A4 P08684 1/20 0.37
KMT2A Q03164 1/20 0.37
DRD1 P21728 2/20 0.36
CHKA P35790 1/20 0.36
HTR1A P08908 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8968431 0.99 ACHE (0.45) ACHEHRH3MAPTNPSR1BCHE
SCHEMBL8970082 0.79 ACHE (0.50) ACHEHRH3MAPTBCHEALDH1A1
SCHEMBL8969676 0.79 ACHE (0.50) ACHEHRH3MAPTBCHEALDH1A1
SCHEMBL8968561 0.78 ACHE (0.63) ACHEMAPTBCHEALDH1A1LMNA
SCHEMBL8969158 0.77 ACHE (0.57) ACHEHRH3MAPTBCHEALDH1A1
SCHEMBL8968341 0.76 ACHE (0.53) ACHEHRH3BCHEALDH1A1LMNA
SCHEMBL8968730 0.76 ACHE (0.63) ACHEHRH3BCHEALDH1A1LMNA
SCHEMBL8970605 0.75 ACHE (0.55) ACHEHRH3MAPTBCHEALDH1A1
SCHEMBL8969839 0.75 ACHE (0.46) ACHEALDH1A1MEN1KMT2A
SCHEMBL8969588 0.75 ACHE (0.55) ACHEHRH3MAPTBCHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
EP-0597956-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1994-05-25 EP disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed