SCHEMBL8968997

SCHEMBL8968997

N=c1c2cc(Br)ccc2nc2n1C1CC3CC(CC2C3)C1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.34
MPO P05164 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ATM Q13315 1/20 0.33
RXFP1 Q9HBX9 2/20 0.33
POLB P06746 1/20 0.33
HTT P42858 2/20 0.33
BCHE P06276 4/20 0.32
ACHE P22303 4/20 0.32
GRIN1 Q05586 4/20 0.32
GRIN2A Q12879 4/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
ADORA1 P30542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8968555 0.90 MPO (0.36) MPOACHE
SCHEMBL8969894 0.85 KDM4E (0.38) BCHEACHEGRIN1GRIN2AADRB2
SCHEMBL8969797 0.84 LRRK2 (0.39) MPOMEN1KMT2AHTTACHE
SCHEMBL8968811 0.81 LRRK2 (0.38)
SCHEMBL8969661 0.77 BCHE (0.34) POLBBCHEACHEGRIN1GRIN2A
SCHEMBL8969460 0.76 ACHE (0.42) MPOPOLBBCHEACHE
SCHEMBL8970437 0.76 MPO (0.36) MPOBCHEACHE
SCHEMBL8968270 0.76
SCHEMBL8968456 0.75 ACHE (0.37) MEN1KMT2APOLBHTTACHE
SCHEMBL8969543 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed