SCHEMBL8968811

SCHEMBL8968811

N=c1c2cc(C(F)(F)F)ccc2nc2n1C1CC3CC(CC2C3)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.38
CYP11B2 P19099 2/20 0.35
CYP11B1 P15538 1/20 0.35
TNF P01375 2/20 0.35
CCNE2 O96020 1/20 0.34
CCNA2 P20248 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
CTSD P07339 1/20 0.33
HTR2B P41595 1/20 0.33
HTR6 P50406 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
KCNH2 Q12809 1/20 0.33
GABBR2 O75899 1/20 0.32
GABBR1 Q9UBS5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969343 0.90 CTSD (0.40) LRRK2CYP11B2CYP11B1TNFHRH3
SCHEMBL8969797 0.81 LRRK2 (0.39) LRRK2
SCHEMBL8970437 0.76 MPO (0.36) LRRK2CYP11B2CYP11B1
SCHEMBL8969661 0.74 BCHE (0.34)
SCHEMBL8969460 0.73 ACHE (0.42) LRRK2
SCHEMBL8969096 0.73 XPO1 (0.36) HRH3CHRNB2CHRNA4KCNH2
SCHEMBL8968456 0.72 ACHE (0.37)
SCHEMBL8969453 0.68 ACHE (0.45) CYP11B2HRH3CHRNB2CHRNA4
SCHEMBL8969422 0.67 HRH4 (0.34)
SCHEMBL8968721 0.67 KDM4E (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed