SCHEMBL8970437

SCHEMBL8970437

N=c1c2ccc(F)cc2nc2n1C1CC3CC(CC2C3)C1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.36
BCHE P06276 4/20 0.35
ACHE P22303 3/20 0.35
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
LRRK2 Q5S007 3/20 0.32
CYP11B2 P19099 3/20 0.32
CYP11B1 P15538 2/20 0.32
CCR3 P51677 1/20 0.32
MAP3K14 Q99558 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969661 0.85 BCHE (0.34) BCHEACHE
SCHEMBL8969460 0.84 ACHE (0.42) MPOBCHEACHELRRK2
SCHEMBL8968555 0.84 MPO (0.36) MPOACHE
SCHEMBL8969437 0.79 BCHE (0.35) BCHEACHE
SCHEMBL8969894 0.77 KDM4E (0.38) BCHEACHE
SCHEMBL8968356 0.77
SCHEMBL8969797 0.76 LRRK2 (0.39) MPOACHELRRK2
SCHEMBL8968811 0.76 LRRK2 (0.38) LRRK2CYP11B2CYP11B1
SCHEMBL8968456 0.75 ACHE (0.37) ACHE
SCHEMBL8969453 0.74 ACHE (0.45) BCHEACHECYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed