SCHEMBL8969644

SCHEMBL8969644

FC(F)(F)c1ccc2c(c1)N=C1C=CC=CN1C2

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSD P07339 8/20 0.44
PNMT P11086 4/20 0.35
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
PARP1 P09874 1/20 0.33
PARP10 Q53GL7 1/20 0.33
TDP2 O95551 1/20 0.33
ADRB1 P08588 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969736 0.89 CTSD (0.34) CTSDPNMTTDP2
SCHEMBL8969486 0.81 MAPK1 (0.34)
SCHEMBL8968478 0.78 ACHE (0.43) CTSDPNMT
SCHEMBL11774305 0.75 CA1 (0.34) CTSD
SCHEMBL8970367 0.74 HTR7 (0.31)
SCHEMBL10767417 0.73 HPGD (0.41) CTSD
SCHEMBL8969612 0.69 PDE3B (0.34)
SCHEMBL8969494 0.69 KDM4E (0.30) PNMT
SCHEMBL8969070 0.69 KDM4E (0.33)
SCHEMBL8969143 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed