SCHEMBL8969736

SCHEMBL8969736

FC(F)(F)c1ccc2c(c1)CN1C=CC=CC1=N2

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSD P07339 7/20 0.34
NOTUM Q6P988 1/20 0.33
PNMT P11086 4/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
ALDH1A1 P00352 1/20 0.31
HRH3 Q9Y5N1 1/20 0.30
TDP2 O95551 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969644 0.89 CTSD (0.44) CTSDPNMTTDP2
SCHEMBL8969494 0.78 KDM4E (0.30) PNMTALDH1A1
SCHEMBL8969612 0.78 PDE3B (0.34) ALDH1A1
SCHEMBL8968669 0.74 NPSR1 (0.31)
SCHEMBL11774305 0.72 CA1 (0.34) CTSD
SCHEMBL8969486 0.72 MAPK1 (0.34) ALDH1A1
SCHEMBL8968478 0.69 ACHE (0.43) CTSDPNMTALDH1A1
SCHEMBL8969002 0.67 ACHE (0.39) ALDH1A1HRH3
SCHEMBL8969143 0.67
SCHEMBL892966 0.66 TDP2 (0.36) NOTUMALDH1A1TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed