SCHEMBL8969704

SCHEMBL8969704

Fc1ccc2c(c1)N=C1C3CC4CC(C3)CC(C4)N1C2

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.36
HTR2B P41595 2/20 0.36
CTSD P07339 7/20 0.34
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33
CHRNA4 P43681 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
MAPK1 P28482 1/20 0.31
HTR6 P50406 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969466 0.85 CTSD (0.49) HTR2CHTR2BCTSD
SCHEMBL8969577 0.84 CTSD (0.34) HTR2CHTR2BCTSDHTR6
SCHEMBL8969760 0.84 CTSD (0.34) CTSD
SCHEMBL8969065 0.83 CTSD (0.51) HTR2CHTR2BCTSDCHRNB2CHRNB4
SCHEMBL9540235 0.80 CTSD (0.47) CTSD
SCHEMBL8968819 0.78 MAPK1 (0.34) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL8969194 0.78 CTSD (0.33) CTSD
SCHEMBL8968314 0.77 PDE3B (0.40) HTR2CHTR2BCTSD
SCHEMBL8969715 0.76
SCHEMBL8968336 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
EP-0597956-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1994-05-25 EP disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed