SCHEMBL8970393

SCHEMBL8970393

COc1cccc2c1CC(CN(CCCN(Cc1ccccc1)S(=O)(=O)c1ccc(F)cc1)Cc1ccccc1)CC2

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 6/20 0.45
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
HTR1A P08908 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
DRD2 P14416 2/20 0.41
KCNA5 P22460 1/20 0.41
KMT2A Q03164 1/20 0.41
BMP1 P13497 1/20 0.41
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969014 0.92 CHRM2 (0.43) TAS2R14CHRM2CHRM1CHRM3HTR1A
SCHEMBL8970649 0.87 BACE1 (0.47) TAS2R14CHRM2CHRM1CHRM3HTR1A
SCHEMBL8970546 0.86 DRD2 (0.43) CHRM2CHRM1CHRM3HTR1ASIGMAR1
SCHEMBL8969348 0.80 MTNR1A (0.46) CHRM2CHRM1CHRM3HTR1ASIGMAR1
SCHEMBL8996694 0.79 MTNR1A (0.46) CHRM2CHRM1CHRM3HTR1ASIGMAR1
SCHEMBL8970412 0.79 CHRM2 (0.48) CHRM2CHRM1CHRM3HTR1ASIGMAR1
SCHEMBL8970549 0.77 MTNR1A (0.54) HTR1ASIGMAR1DRD2
SCHEMBL8971881 0.76 CA1 (0.44) HTR1ASIGMAR1DRD2
SCHEMBL8970432 0.73 CHRM2 (0.48) CHRM2CHRM1CHRM3KMT2A
SCHEMBL8970496 0.72 CHRM2 (0.48) CHRM2CHRM1CHRM3DRD2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585392-A TREATING OR PREVENTING STROKES BAYER AKTIENGESELLSCHAFT (DE) 1996-12-17 US disclosed
US-5506246-A Method for treating depression using substituted aminomethyltetralins and their heterocyclic analogues BAYER AKTIENGESELLSCHAFT (DE) 1996-04-09 US disclosed
EP-0352613-B1 Substituted amino methyl tetralines, and their heterocyclic analogous compounds BAYER AG (DE) 1994-04-20 EP disclosed
US-5300523-A Binding serotonin receptors, treating nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1994-04-05 US disclosed
US-5137901-A For binding 5-HT 1 receptors; treating central nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1992-08-11 US disclosed
EP-0352613-A2 Substituted amino methyl tetralines, and their heterocyclic analogous compounds BAYER AG (DE) 1990-01-31 EP disclosed