SCHEMBL8971881

SCHEMBL8971881

CCOC(=O)NCCCN(Cc1ccccc1)CC1CCc2cccc(OC)c2C1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ACHE P22303 1/20 0.44
MTNR1A P48039 4/20 0.43
MTNR1B P49286 4/20 0.43
DRD2 P14416 3/20 0.43
HTR1A P08908 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
CYP1A2 P05177 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALOX15 P16050 1/20 0.42
DRD3 P35462 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8970549 0.88 MTNR1A (0.54) MTNR1AMTNR1BDRD2HTR1ASIGMAR1
SCHEMBL8969348 0.81 MTNR1A (0.46) MTNR1AMTNR1BDRD2HTR1ASIGMAR1
SCHEMBL8996694 0.80 MTNR1A (0.46) CA1CA2ACHEMTNR1AMTNR1B
SCHEMBL8972304 0.80 MTNR1A (0.49) CA1CA2ACHEMTNR1AMTNR1B
SCHEMBL8970546 0.78 DRD2 (0.43) DRD2HTR1ASIGMAR1DRD3
SCHEMBL8970393 0.76 TAS2R14 (0.45) DRD2HTR1ASIGMAR1
SCHEMBL8969014 0.74 CHRM2 (0.43) DRD2HTR1ASIGMAR1
SCHEMBL8969631 0.74 MTNR1A (0.51) MTNR1AMTNR1BDRD2HTR1ASIGMAR1
SCHEMBL9241035 0.73 MTNR1A (0.60) MTNR1AMTNR1BDRD2CYP1A2MAPT
Hydrochloric Acid SCHEMBL9242384 0.72 MTNR1A (0.59) MTNR1AMTNR1BDRD2CYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585392-A TREATING OR PREVENTING STROKES BAYER AKTIENGESELLSCHAFT (DE) 1996-12-17 US disclosed
US-5506246-A Method for treating depression using substituted aminomethyltetralins and their heterocyclic analogues BAYER AKTIENGESELLSCHAFT (DE) 1996-04-09 US disclosed
EP-0352613-B1 Substituted amino methyl tetralines, and their heterocyclic analogous compounds BAYER AG (DE) 1994-04-20 EP disclosed
US-5300523-A Binding serotonin receptors, treating nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1994-04-05 US disclosed
US-5137901-A For binding 5-HT 1 receptors; treating central nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1992-08-11 US disclosed
EP-0352613-A2 Substituted amino methyl tetralines, and their heterocyclic analogous compounds BAYER AG (DE) 1990-01-31 EP disclosed