SCHEMBL8970415

SCHEMBL8970415

NC(=O)c1cccc(C(=O)n2c3ccc2c(Cl)c3)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.47
ROCK2 O75116 1/20 0.40
PIM1 P11309 1/20 0.40
PIM3 Q86V86 1/20 0.40
TTK P33981 1/20 0.39
MAP2K4 P45985 1/20 0.39
GAA P10253 2/20 0.37
MGAM O43451 1/20 0.37
AMY1A P0DUB6 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
PARP15 Q460N3 2/20 0.37
PARP10 Q53GL7 2/20 0.37
CNR1 P21554 1/20 0.37
TSHR P16473 1/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
ELANE P08246 1/20 0.36
PIK3R2 O00459 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366924 0.86 PARP1 (0.40) PARP1ROCK2PIM1PIM3PARP15
SCHEMBL29120355 0.84 PARP1 (0.39) PARP1ROCK2PIM1PIM3PARP15
SCHEMBL4434522 0.81 PARP1 (0.52) PARP1GAAPARP15PARP10TSHR
Terephthalamide SCHEMBL11492620 0.79 PARP1 (0.47) PARP1ROCK2PIM1PIM3TTK
SCHEMBL8855118 0.75 DHODH (0.45) PARP1TSHRMEN1MAPTKMT2A
SCHEMBL10707481 0.74 LMNA (0.57) PARP1MEN1MAPTKMT2AELANE
Terephthalamide SCHEMBL11494225 0.72 MAPT (0.58) PARP1PARP15PARP10TSHRMEN1
SCHEMBL31021028 0.71 PARP1 (0.73) PARP1PARP15PARP10TSHRMEN1
SCHEMBL36694 0.71 PARP1 (0.73) PARP1PARP15PARP10TSHRMEN1
Water SCHEMBL7768285 0.69 PARP1 (0.70) PARP1PARP15PARP10TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0502953-B1 QUATERNARY AMMONIUM POLYARYLAMIDES DU PONT (US) 1996-02-07 EP claimed
US-5242991-A Electronic circuits and molding materials E. I. DU PONT DE NEMOURS AND COMPANY (US) 1993-09-07 US claimed
EP-0502953-A1 QUATERNARY AMMONIUM POLYARYLAMIDES. DU PONT (US) 1992-09-16 EP claimed
WO-1991008248-A1 QUATERNARY AMMONIUM POLYARYLAMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1991-06-13 WO claimed
US-5407626-A Deprotenation of the amide N by reacting with a quaternary amine to form an anionic polymer; casting from solution; desolventizing; heating to alkylate or neutralize E. I. DU PONT DE NEMOURS AND COMPANY (US) 1995-04-18 US disclosed
US-5242991-A Electronic circuits and molding materials E. I. DU PONT DE NEMOURS AND COMPANY (US) 1993-09-07 US disclosed