SCHEMBL8972154

SCHEMBL8972154

O=C[C@H]1CC[C@H](c2ccc(Cl)c(F)c2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 5/20 0.35
SLC6A4 P31645 4/20 0.35
SLC6A3 Q01959 4/20 0.35
RIPK1 Q13546 1/20 0.35
HTR7 P34969 1/20 0.34
HSD11B1 P28845 1/20 0.34
KCNH2 Q12809 3/20 0.33
CYP2D6 P10635 2/20 0.33
PANK3 Q9H999 1/20 0.33
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
KCNJ8 Q15842 1/20 0.32
MAPK14 Q16539 1/20 0.32
PIM1 P11309 1/20 0.32
CSNK2A2 P19784 1/20 0.32
CSNK2B P67870 1/20 0.32
PIM3 Q86V86 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
CHRNA3 P32297 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9311759 1.00 SLC6A2 (0.35) SLC6A2SLC6A4SLC6A3RIPK1HTR7
SCHEMBL9313677 0.92 OPRL1 (0.36) HSD11B1PANK3ESR2PTGIRPTGDR
SCHEMBL8517594 0.92 OPRL1 (0.36) HSD11B1PANK3ESR2PTGIRPTGDR
SCHEMBL28710880 0.87 CYP2D6 (0.46) SLC6A2SLC6A4SLC6A3HTR7KCNH2
SCHEMBL15517006 0.86 SLC6A3 (0.42) SLC6A2SLC6A4SLC6A3RIPK1HTR7
SCHEMBL6455890 0.86 RIPK1 (0.32) SLC6A2SLC6A4SLC6A3RIPK1HTR7
SCHEMBL6455888 0.86 RIPK1 (0.32) SLC6A2SLC6A4SLC6A3RIPK1HTR7
SCHEMBL4931479 0.85 USP30 (0.38) ESR2
SCHEMBL4931475 0.85 USP30 (0.38) ESR2
SCHEMBL8962617 0.83 SLC6A2 (0.35) SLC6A2SLC6A4SLC6A3RIPK1HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433836-B1 Halophenyl substituted dioxanes HOFFMANN LA ROCHE (CH) 1996-03-27 EP disclosed
US-5322638-A Halophenyl substituted dioxanes HOFFMANN-LA ROCHE INC. (US) 1994-06-21 US disclosed
EP-0433836-A2 Halophenyl substituted dioxanes F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed