SCHEMBL8973600

SCHEMBL8973600

O=C1CN(S(=O)(=O)c2cc3cc(Br)ccc3o2)C(=O)N1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.43
CA12 O43570 2/20 0.43
CA9 Q16790 2/20 0.43
CA1 P00915 1/20 0.43
CYP2A6 P11509 1/20 0.38
LMNA P02545 4/20 0.38
PKM P14618 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HPGD P15428 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GPR35 Q9HC97 1/20 0.38
RAB9A P51151 4/20 0.38
ALDH1A1 P00352 3/20 0.38
NPC1 O15118 3/20 0.38
PIM1 P11309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9000148 0.90 MAOB (0.35) CA2CA12CA9CA1PKM
SCHEMBL8800240 0.85 AKR1B1 (0.47) CA2CA12CA9CA1MEN1
SCHEMBL8800132 0.83 CA2 (0.49) CA2CA12CA9CA1MEN1
SCHEMBL8799877 0.79 MEN1 (0.33) MEN1KMT2AALDH1A1MAPT
SCHEMBL8798817 0.76 TERT (0.34) CA2MEN1KMT2AALDH1A1MAPT
SCHEMBL8973637 0.76 MMP2 (0.46) PKMMEN1KMT2AALDH1A1MAPT
SCHEMBL9000112 0.73 MEN1 (0.36) MEN1KMT2AALDH1A1MAPT
SCHEMBL8799930 0.73 MEN1 (0.35) PKMMEN1KMT2AALDH1A1MAPT
SCHEMBL10679786 0.72 MEN1 (0.39) MEN1KMT2AALDH1A1MAPTSMN1; SMN2
SCHEMBL8799255 0.72 CA2 (0.46) CA2CA12CA9CA1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0444546-B1 Hydantoin derivatives for use as hypoglycemic and/or hypolipidemic agents MOCHIDA PHARM CO LTD (JP) 1996-09-11 EP disclosed
US-RE35279-E ALDOSE REDUCTASE INHIBITORS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
US-5202339-A Hypoglycemic, hypolipedemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1993-04-13 US disclosed
WO-1991012803-A1 HYDANTOIN DERIVATIVES FOR USE AS HYPOGLYCEMIC AND/OR HYPOLIPIDEMIC AGENTS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-09-05 WO disclosed
EP-0444546-A1 Hydantoin derivatives for use as hypoglycemic and/or hypolipidemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-09-04 EP disclosed
US-5004751-A Antidiabetic agents; aldoe reductase inhibitors MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-04-02 US disclosed
US-4914099-A TREATMENT OR PREVENTION OF DIABETIC COMPLICATIONS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-04-03 US disclosed
WO-1990002126-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-03-08 WO disclosed
EP-0355827-A2 Hydantoin derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-02-28 EP disclosed
WO-1989001934-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-09 WO disclosed
EP-0305947-A1 Hydantoin derivatives, process for their preparation and pharmaceutical compositions containing the same as well as their use MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-08 EP disclosed