SCHEMBL8973733

SCHEMBL8973733

NS(=O)(=O)c1ccc(C2=CC(C(F)(F)F)(C(F)(F)F)C=C2c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.68
PTGS2 P35354 7/20 0.56
PTGS1 P23219 3/20 0.56
CA12 O43570 4/20 0.49
CA2 P00918 4/20 0.49
CA9 Q16790 4/20 0.49
CA1 P00915 2/20 0.49
MAPT P10636 1/20 0.49
CYP2C9 P11712 1/20 0.47
PDPK1 O15530 1/20 0.46
CHRNA7 P36544 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974490 0.87 CA2 (0.50) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974255 0.86 PTGS1 (0.53) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974616 0.86 KIF11 (0.70) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974399 0.86 KIF11 (0.50) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974073 0.86 KIF11 (0.50) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974655 0.85 PTGS2 (0.56) KIF11PTGS2PTGS1
SCHEMBL8974169 0.85 CA2 (0.55) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974123 0.85 KIF11 (0.68) KIF11PTGS2PTGS1CA12CA2
SCHEMBL9117080 0.84 KIF11 (0.66) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974138 0.83 KIF11 (0.45) KIF11PTGS2PTGS1CA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed