SCHEMBL8974255

SCHEMBL8974255

NS(=O)(=O)c1ccc(C2=CC(C(F)(F)F)(C(F)(F)F)C=C2c2ccc(F)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 14/20 0.53
PTGS2 P35354 14/20 0.53
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
KIF11 P52732 2/20 0.47
SOS1 Q07889 1/20 0.47
CA2 P00918 2/20 0.46
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46
CA1 P00915 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974169 0.86 CA2 (0.55) PTGS1PTGS2MAOAMAOBKIF11
SCHEMBL8973733 0.86 KIF11 (0.68) PTGS1PTGS2KIF11CA2CA12
SCHEMBL8973770 0.86 CA2 (0.41) PTGS1PTGS2MAOAMAOBCA2
SCHEMBL8975948 0.86 CA2 (0.41) PTGS1PTGS2MAOAMAOBKIF11
SCHEMBL8974490 0.85 CA2 (0.50) PTGS1PTGS2KIF11CA2CA12
SCHEMBL8973922 0.84 PTGS2 (0.66) PTGS1PTGS2
SCHEMBL8974555 0.83 KIF11 (0.41) PTGS1PTGS2MAOAMAOBKIF11
SCHEMBL8973874 0.82 PTGS2 (0.57) PTGS1PTGS2MAOAMAOBSOS1
SCHEMBL8974138 0.81 KIF11 (0.45) PTGS1PTGS2KIF11CA2CA12
SCHEMBL214628 0.81 PTGS2 (0.56) PTGS1PTGS2MAOAMAOBSOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed