SCHEMBL8974113

SCHEMBL8974113

COc1ccc(C2=CCC=C2c2ccc(S(N)(=O)=O)cc2)cc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.46
PTGS1 P23219 15/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
KIF11 P52732 1/20 0.45
S1PR1 P21453 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974106 0.89 PTGS2 (0.48) PTGS2PTGS1KIF11
SCHEMBL9117719 0.85 PTGS2 (0.56) PTGS2PTGS1CA12CA1CA2
SCHEMBL8974584 0.84 KIF11 (0.55) PTGS2PTGS1CA12CA1CA2
SCHEMBL8974532 0.84 KIF11 (0.48) PTGS2PTGS1CA12CA1CA2
SCHEMBL8974267 0.84 PTGS2 (0.66) PTGS2PTGS1
Benzenesulfonamide SCHEMBL9117409 0.83 PTGS2 (0.40) PTGS2PTGS1CA12CA1CA2
SCHEMBL8974152 0.82 KIF11 (0.56) PTGS2PTGS1CA12CA2CA9
SCHEMBL8974164 0.82 PTGS2 (0.61) PTGS2PTGS1CA12CA1CA2
SCHEMBL8974570 0.81 PTGS2 (0.57) PTGS2PTGS1CA1CA2CA9
SCHEMBL8973775 0.81 KIF11 (0.51) PTGS2PTGS1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed