SCHEMBL8974115

SCHEMBL8974115

CS(=O)(=O)c1ccc(C2=CC(C(=O)O)(C(=O)O)C=C2c2ccc(C(F)(F)F)cc2)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.40
PPARD Q03181 3/20 0.38
MAP4K4 O95819 2/20 0.38
CTSK P43235 1/20 0.38
PTGS2 P35354 3/20 0.36
PTGS1 P23219 1/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36
MMP9 P14780 1/20 0.36
MMP13 P45452 1/20 0.36
PIK3CA P42336 1/20 0.36
KCNH2 Q12809 1/20 0.36
MINK1 Q8N4C8 1/20 0.36
PI4KB Q9UBF8 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
KIF11 P52732 1/20 0.35
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973759 0.88 POLB (0.41) POLBPPARDMAP4K4CTSKPTGS2
SCHEMBL8973844 0.88 KIF11 (0.40) POLBPPARDMAP4K4PTGS2PTGS1
SCHEMBL8974628 0.86 PTGS2 (0.43) POLBMAP4K4CTSKPTGS2PTGS1
SCHEMBL8974809 0.86 PTGS2 (0.40) POLBPPARDMAP4K4CTSKPTGS2
SCHEMBL8973745 0.85 POLB (0.39) POLBMAP4K4CTSKPTGS2PIK3CA
SCHEMBL8974352 0.84 POLB (0.38) POLBMAP4K4CTSKPTGS2PIK3CA
SCHEMBL9118890 0.83 PTGS2 (0.48) POLBMAP4K4CTSKPTGS2PTGS1
SCHEMBL9119094 0.82 POLB (0.38) POLBMAP4K4CTSKPTGS2PTGS1
SCHEMBL8974615 0.82 POLB (0.40) POLBMAP4K4CTSKPTGS2PTGS1
SCHEMBL8974707 0.81 PPARD (0.38) POLBPPARDMAP4K4CTSKPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed