SCHEMBL8974144

SCHEMBL8974144

COC(=O)C1C=C(c2ccc(C(F)(F)F)cc2)C(c2ccc(S(N)(=O)=O)cn2)=C1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.44
CA2 P00918 5/20 0.41
CA12 O43570 3/20 0.41
CA1 P00915 3/20 0.41
CA9 Q16790 3/20 0.41
MAPT P10636 1/20 0.41
CA4 P22748 2/20 0.40
CA7 P43166 2/20 0.40
PTGS2 P35354 5/20 0.39
PTGS1 P23219 2/20 0.39
GAA P10253 2/20 0.38
KDM4E B2RXH2 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CHRNA7 P36544 2/20 0.37
GCK P35557 1/20 0.36
GCKR Q14397 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973885 0.94 KIF11 (0.46) KIF11CA2CA12CA1CA9
SCHEMBL8974718 0.92 PTGS2 (0.39) KIF11PTGS2PTGS1GAA
SCHEMBL8974768 0.88 KIF11 (0.47) KIF11CA2CA12CA1CA9
SCHEMBL8974416 0.88 CA2 (0.41) CA2CA12CA1CA9CA4
SCHEMBL8974201 0.88 KIF11 (0.57) KIF11CA2CA12CA1CA9
SCHEMBL8974486 0.88 PTGS2 (0.42) KIF11PTGS2PTGS1
SCHEMBL8974632 0.85 KIF11 (0.50) KIF11CA2CA12CA1CA9
SCHEMBL8974507 0.84 PTGS2 (0.41) CA2CA12CA1CA9CA4
SCHEMBL8974121 0.83 KIF11 (0.51) KIF11CA2CA12CA1CA9
SCHEMBL8974153 0.83 KIF11 (0.40) KIF11CA2CA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed