SCHEMBL8974176

SCHEMBL8974176

CCc1ccc(C2=CCC=C2c2ccc(S(N)(=O)=O)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 14/20 0.68
PTGS1 P23219 2/20 0.48
PTGS2 P35354 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
CA12 O43570 9/20 0.47
CA9 Q16790 8/20 0.47
CA1 P00915 8/20 0.46
CA14 Q9ULX7 6/20 0.46
CA7 P43166 4/20 0.46
CA4 P22748 3/20 0.46
CA6 P23280 3/20 0.46
CA5A P35218 3/20 0.46
CA5B Q9Y2D0 3/20 0.46
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
GLA P06280 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974175 0.85 PTGS2 (0.47) CA2PTGS1PTGS2UCHL1
SCHEMBL23512338 0.84 CA2 (0.88) CA2PTGS1PTGS2SMN1; SMN2CA12
SCHEMBL8974562 0.84 CA2 (0.68) CA2PTGS2SMN1; SMN2CA12CA9
SCHEMBL8974202 0.83 CA2 (0.50) CA2PTGS1PTGS2CA12CA9
SCHEMBL635526 0.82 CA2 (1.00) CA2SMN1; SMN2CA12CA9CA1
SCHEMBL8974305 0.81 CA2 (0.64) CA2PTGS1PTGS2CA12CA9
SCHEMBL8974243 0.80 CA2 (0.71) CA2PTGS1PTGS2CA12CA9
SCHEMBL8974782 0.80 CA2 (0.68) CA2PTGS1PTGS2CA12CA9
SCHEMBL8974406 0.78 PTGS2 (0.60) CA2PTGS1PTGS2CA12CA9
SCHEMBL8973815 0.78 CA2 (0.52) CA2PTGS1PTGS2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed